SR9011 as an agonist of Rev-ErbAα with a half-maximum inhibitory concentration (IC50) = 790 nM for Rev-Erbα and IC50 = 560 nM for Rev-ErbAβ. It has been used in the study of the regulation of the circadian rhythm and its links to immune system function, inflammation and cancer.
SR9011 VS SR9009
SR 9011 was developed to improve the poor bioavailability, short half-life and frequent repeated dosing issues of SR9009. The improved bioavailability of SR 9011 means that it is more effectively absorbed and utilized by the body when taken orally compared to SR9009.
SR9011 Benefits
Increased endurance
Lower body fat
Decreased anxiety and inflammation
Increased muscle mass
SR9011 dosage for bodybuilding
Although there is no FDA-established dosage for SR9011, most users recommend starting with around 10 mg per day. The recommended dosages for different experience levels are:
– Beginner: 10 mg per day
– Intermediate: 20 mg per day
– Advanced: 30+ mg per day
The half-life of SR 9011 is around 4 hours, so it’s advised to split the dosage into three parts and take it in the morning, noon, and evening to maintain optimal levels throughout the day. Most users take between 15 and 30 mg per day, divided into three doses.
SR9011 Side Effects
As of now, the only known side effect of SR9011 is wakefulness. However, the compound is not well-researched yet, which means it could potentially have other side effects that are not yet known.
SR9011 Chemical Properties
Boiling point 642.8±50.0 °C(Predicted)
density 1.254±0.06 g/cm3(Predicted)
storage temp. Keep in dark place,Sealed in dry,Store in freezer, under -20°C
solubility Chloroform (Slightly), Methanol (Slightly)
form Solid
pka 14.71±0.40(Predicted)
color Dark Yellow to Very Dark Brown
InChI InChI=1S/C23H31ClN4O3S/c1-2-3-4-12-25-23(29)27-13-11-19(16-27)15-26(14-18-5-7-20(24)8-6-18)17-21-9-10-22(32-21)28(30)31/h5-10,19H,2-4,11-17H2,1H3,(H,25,29)
InChIKey PPUYOYQTTWJTIU-UHFFFAOYSA-N
SMILES N1(C(NCCCCC)=O)CCC(CN(CC2=CC=C(Cl)C=C2)CC2SC([N+]([O-])=O)=CC=2)C1
More Introduction:https://en.wikipedia.org/wiki/SR9011
